Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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X139028-1g | 1g | In stock | $12.90 | |
X139028-5g | 5g | In stock | $48.90 | |
X139028-10g | 10g | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $87.90 | |
X139028-25g | 25g | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $144.90 | |
X139028-100g | 100g | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $519.90 |
Platelet COX inhibitor
Synonyms | sulfinpyrazone|57-96-5|Sulphinpyrazone|Anturane|(+/-)-SULFINPYRAZONE|Sulfinpyrazon|Anturan|Diphenylpyrazone|Sulfoxyphenylpyrazolidine|Anturanil|Anturidin|Enturen|Anturano|1,2-Diphenyl-4-(2-(phenylsulfinyl)ethyl)pyrazolidine-3,5-dione|USAF GE-13|Sulfinpyra |
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Specifications & Purity | ≥96% |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Action Type | ANTAGONIST, INHIBITOR |
Mechanism of action | Antagonist of FPR1;Inhibitor of Urate anion exchanger 1 |
Product Description | Product Describtion: Sulfinpyrazone is a free radical scavenger that is an inhibitor of organic anion transporters (OATP) and is an effective uricosuric chemical. It is a proposed nonselective UGT (UDP-glucuronosyltransferases) inhibitor. The transport of sulfinpyrazone in MDCKII-MRP1 cells is associated with GSH export, except in high concentrations, and is a substrate for MRP2 (multidrug resistance protein). Product Application: cleaning products,cosmetics,food and beverages,forensics and toxicology,personal care,pharmaceutical (small molecule),veterinary |
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IUPAC Name | 4-[2-(benzenesulfinyl)ethyl]-1,2-diphenylpyrazolidine-3,5-dione |
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INCHI | InChI=1S/C23H20N2O3S/c26-22-21(16-17-29(28)20-14-8-3-9-15-20)23(27)25(19-12-6-2-7-13-19)24(22)18-10-4-1-5-11-18/h1-15,21H,16-17H2 |
InChi Key | MBGGBVCUIVRRBF-UHFFFAOYSA-N |
Canonical SMILES | C1=CC=C(C=C1)N2C(=O)C(C(=O)N2C3=CC=CC=C3)CCS(=O)C4=CC=CC=C4 |
Isomeric SMILES | C1=CC=C(C=C1)N2C(=O)C(C(=O)N2C3=CC=CC=C3)CCS(=O)C4=CC=CC=C4 |
WGK Germany | 3 |
RTECS | UQ8575000 |
PubChem CID | 5342 |
Molecular Weight | 404.48 |
CAS Registry No. | 57-96-5 |
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Wikipedia | Sulfinpyrazone |
PubChem CID | 5342 |
ChEMBL Ligand | CHEMBL832 |
DrugBank Ligand | DB01138 |
DrugCentral Ligand | 2528 |
GPCRdb Ligand | sufinpyrazone |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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F2224204 | Certificate of Analysis | Apr 03, 2024 | X139028 |
F2224205 | Certificate of Analysis | Apr 03, 2024 | X139028 |
F2224243 | Certificate of Analysis | Apr 03, 2024 | X139028 |
F2428071 | Certificate of Analysis | Apr 03, 2024 | X139028 |
X139028-5g;G2010049 | Certificate of Analysis | May 07, 2022 | X139028 |
X139028-1g;G2010048 | Certificate of Analysis | May 07, 2022 | X139028 |
Solubility | Slightly soluble in water; Soluble in Acetone,Chloroform; Slightly soluble in Alcohol,Ether |
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Melt Point(°C) | 131 °C |
Pictogram(s) | GHS07 |
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Signal | Warning |
Hazard Statements | H302:Harmful if swallowed |
Precautionary Statements | P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P330:Rinse mouth. P301+P317:IF SWALLOWED: Get medical help. |
WGK Germany | 3 |
RTECS | UQ8575000 |
Merck Index | 8949 |