TPMPA - ≥98%(HPLC), high purity , CAS No.182485-36-5, Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit

Item Number

T287271

• Synonyms: TPMPA|182485-36-5|methyl(1,2,3,6-tetrahydropyridin-4-yl)phosphinic acid|Tpmpa [MI]|Phosphinic acid, P-methyl-P-(1,2,3,6-tetrahydro-4-pyridinyl)-|(1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid|CHEMBL397209|TR7I0800L2|P-Methyl-P-(1,2,3,6-tetrahydro-4
• Specifications & Purity: Moligand™, ≥98%(HPLC)
• Biochemical and Physiological Mechanisms: A selective, competitive GABAA-ρantagonist with only minimal effects on GABAAand GABABreceptors (Kbvalues are 2.1μM (antagonist), 320μM (antagonist) and EC50~ 500μM (weak agonist) respectively). Displays 8-fold selectivity for human recombinantρ1 receptor
• Storage Temp: Room temperature
• Shipped In: Normal
• Grade: Moligand™
• Action Type: ANTAGONIST
• Mechanism of action: Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit