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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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Z288507-5mg | 5mg | In stock | $137.90 | |
Z288507-10mg | 10mg | In stock | $226.90 | |
Z288507-25mg | 25mg | In stock | $503.90 | |
Z288507-50mg | 50mg | In stock | $939.90 | |
Z288507-100mg | 100mg | In stock | $1,583.90 |
CaV3.x blocker
Synonyms | 1199236-64-0|Z944|Ulixacaltamide|Z 944|N-((1-(2-(tert-Butylamino)-2-oxoethyl)piperidin-4-yl)methyl)-3-chloro-5-fluorobenzamide|Ulixacaltamide [INN]|Z-944|QT2PJH89C3|N-[[1-[2-(tert-butylamino)-2-oxoethyl]piperidin-4-yl]methyl]-3-chloro-5-fluorobenzamide|CH |
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Specifications & Purity | ≥98%(HPLC) |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Grade | Moligand™ |
Action Type | CHANNEL BLOCKER |
Mechanism of action | Channel blocker of Ca v3.1;Channel blocker of Ca v3.2;Channel blocker of Ca v3.3 |
Product Description | Product Introduction Z944 is a T-type calcium channel blocker. Z944 delays the progression of seizures in the amygdala kindling model. Z944 disrupts prepulse inhibition in both epileptic and non-epileptic rats. |
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IUPAC Name | N-[[1-[2-(tert-butylamino)-2-oxoethyl]piperidin-4-yl]methyl]-3-chloro-5-fluorobenzamide |
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INCHI | InChI=1S/C19H27ClFN3O2/c1-19(2,3)23-17(25)12-24-6-4-13(5-7-24)11-22-18(26)14-8-15(20)10-16(21)9-14/h8-10,13H,4-7,11-12H2,1-3H3,(H,22,26)(H,23,25) |
InChi Key | JOCLITFYIMJMNK-UHFFFAOYSA-N |
Canonical SMILES | CC(C)(C)NC(=O)CN1CCC(CC1)CNC(=O)C2=CC(=CC(=C2)Cl)F |
Isomeric SMILES | CC(C)(C)NC(=O)CN1CCC(CC1)CNC(=O)C2=CC(=CC(=C2)Cl)F |
PubChem CID | 44540045 |
Molecular Weight | 383.89 |
PubChem CID | 44540045 |
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CAS Registry No. | 1199236-64-0 |
RCSB PDB Ligand | DZR |
Enter Lot Number to search for COA:
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Lot Number | Certificate Type | Date | Item |
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I2222239 | Certificate of Analysis | Jul 13, 2022 | Z288507 |
I2222240 | Certificate of Analysis | Jul 13, 2022 | Z288507 |
I2222241 | Certificate of Analysis | Jul 13, 2022 | Z288507 |
I2222242 | Certificate of Analysis | Jul 13, 2022 | Z288507 |
I2222243 | Certificate of Analysis | Jul 13, 2022 | Z288507 |
Solubility | Solvent:DMSO, Max Conc. mg/mL: 38.39, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 38.39, Max Conc. mM: 100 |
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Melt Point(°C) | 122-124°C |