Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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Z127987-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $89.90 | |
Z127987-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $139.90 | |
Z127987-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $299.90 | |
Z127987-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $499.90 | |
Z127987-100mg | 100mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $899.90 |
PDE3/4 inhibitor
Synonyms | 6-(4-Difluoromethoxy-3-methoxyphenyl)-3(2H)-pyridazinone |
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Specifications & Purity | ≥98% |
Biochemical and Physiological Mechanisms | Phosphodiesterase inhibitor, selective for PDE3 and 4 (IC50values are 0.5 and 0.8μM respectively). |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Product Description | Zardaverine is a newly developed dual-selective PDE3/4 inhibitor with IC50 values of 0.5 uM and 0.8 uM respectively. |
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IUPAC Name | 3-[4-(difluoromethoxy)-3-methoxyphenyl]-1H-pyridazin-6-one |
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INCHI | InChI=1S/C12H10F2N2O3/c1-18-10-6-7(2-4-9(10)19-12(13)14)8-3-5-11(17)16-15-8/h2-6,12H,1H3,(H,16,17) |
InChi Key | HJMQDJPMQIHLPB-UHFFFAOYSA-N |
Canonical SMILES | COC1=C(C=CC(=C1)C2=NNC(=O)C=C2)OC(F)F |
Isomeric SMILES | COC1=C(C=CC(=C1)C2=NNC(=O)C=C2)OC(F)F |
PubChem CID | 5723 |
Molecular Weight | 268.22 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
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J2412798 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412799 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412800 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412801 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412802 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412803 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412804 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
J2412805 | Certificate of Analysis | Sep 30, 2024 | Z127987 |
Solubility | Solvent:DMSO, Max Conc. mg/mL: None, Max Conc. mM: 100 |
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