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ZM 241385 - ≥99%, high purity , CAS No.139180-30-6, Antagonist of A 1 receptor;Antagonist of A 2A receptor;Antagonist of A 2B receptor;Antagonist of A 3 receptor

Specifications & Purity:  ≥99%
Item Number
Z275221
Grouped product items
SKUSizeAvailabilityPrice Qty
Z275221-10mg
10mg
In stock
$107.90
Z275221-25mg
25mg
In stock
$243.90
Z275221-50mg
50mg
In stock
$391.90
Z275221-100mg
100mg
In stock
$608.90
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Potent, selective A 2A antagonist

View related series
A1 receptor Antagonist A2A receptor Antagonist A2B receptor Antagonist A3 receptor Antagonist

Basic Description

Synonyms139180-30-6|ZM241385|ZM 241385|ZM-241385|4-(2-((7-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino)ethyl)phenol|4-(2-[7-Amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol|5NIC36BO71|CHEMBL113142|ZM-241,385|C16
Specifications & Purity≥99%
Storage TempStore at -20°C
Shipped InDry ice
Action TypeANTAGONIST
Mechanism of actionAntagonist of A 1 receptor;Antagonist of A 2A receptor;Antagonist of A 2B receptor;Antagonist of A 3 receptor

Associated Targets

ADORA2A Tclin Adenosine receptor A2a 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

ADORA2B Tclin Adenosine receptor A2b 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

ADORA1 Tclin Adenosine receptor A1 0 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

ADORA3 Tchem Adenosine receptor A3 1 Activities

Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

IUPAC Name 4-[2-[[7-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]amino]ethyl]phenol
INCHI InChI=1S/C16H15N7O2/c17-14-20-15(18-8-7-10-3-5-11(24)6-4-10)21-16-19-13(22-23(14)16)12-2-1-9-25-12/h1-6,9,24H,7-8H2,(H3,17,18,19,20,21,22)
InChi Key PWTBZOIUWZOPFT-UHFFFAOYSA-N
Canonical SMILES C1=COC(=C1)C2=NN3C(=NC(=NC3=N2)NCCC4=CC=C(C=C4)O)N
Isomeric SMILES C1=COC(=C1)C2=NN3C(=NC(=NC3=N2)NCCC4=CC=C(C=C4)O)N
PubChem CID 176407
Molecular Weight 337.34

Certificates

Certificate of Analysis(COA)

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To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section

4 results found

Lot NumberCertificate TypeDateItem
I2202929Certificate of AnalysisJun 13, 2023 Z275221
I2202931Certificate of AnalysisJun 13, 2023 Z275221
I2202932Certificate of AnalysisJun 05, 2023 Z275221
I2202930Certificate of AnalysisJun 05, 2023 Z275221

Chemical and Physical Properties

SolubilitySoluble in DMSO to 100 mM and in ethanol to 5 mM (with warming)

Safety and Hazards(GHS)

Pictogram(s) GHS06
Signal Danger
Hazard Statements H301
Precautionary Statements P321,P405,P501,P264,P270,P330,P301+P316

Related Documents

 SDS

 Specification Sheet

References

1. Basu M et al..  (2020)  Increased host ATP efflux and its conversion to extracellular adenosine is crucial for establishing Leishmania infection..  J Cell Sci,  133  (7):   [PMID:32079656]

Solution Calculators

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